Drug & chemical–disease

ChEMBL

Bioactive small molecules
"The open bioactivity database — small molecules and their assayed targets."
bioactivitytargetsopen

About the resource

ChEMBL is EMBL-EBI's manually curated open bioactivity database. It captures bioactivity measurements (IC50, EC50, Ki, Kd and similar) from medicinal-chemistry journals and selected high-throughput datasets, plus extensive drug, mechanism, indication and approval metadata. The current release contains over 2 million compounds, 20 million bioactivity measurements and around 15,000 targets, including disease- and pathway-context information for many drugs.

ChEMBL is the open foundation behind much of cheminformatics: it underpins Open Targets prioritisation, dozens of QSAR and ML models, drug-repurposing efforts and target-discovery pipelines. CC BY-SA 3.0.

What you'd use it for

  1. 01Pull bioactivity data for a target across compounds and assays
  2. 02Build a QSAR / ML model on disease-relevant chemistry
  3. 03Audit a drug's mechanism, indications and approval status
  4. 04Power target-discovery analyses against open bioactivity evidence

How you access it

Web UIREST APIFTP downloads (SQLite, MySQL, ChEMBL_RDF)

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